A stable analog of PGF2α 2-glyceryl ester incorporating an activity-enhancing 17-phenyl substitution

17-phenyl trinor Prostaglandin F2α serinol amide – 10 mg

Brand:
Cayman
CAS:
1175838-84-2
Storage:
-20
UN-No:
De Minimis - 1170 / 3

2-Arachidonyl glycerol (2-AG) exhibits cannabinoid agonist activity at the central cannabinoid (CB1) receptor, is an important endogenous monoglyceride species, and is thus considered to be the natural ligand for the CB1 receptor{5306,6819}. 2-AG can also be metabolized by COX-2 to form prostaglandin (PG) 2-glyceryl esters.{11045} These 2-glyceryl esters rapidly equilibrate to form 90:10 mixtures favoring the more stable 1-glyceryl ester. 17-phenyl trinor PGF2α serinol amide is a stable analog of PGF2α 2-glyceryl ester incorporating an activity-enhancing 17-phenyl substitution. The biological activity of 17-phenyl trinor PGF2α serinol amide has not yet been determined.  

 

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SKU: 10004237 - 10 mg Category:

Description

A stable analog of PGF2α 2-glyceryl ester incorporating an activity-enhancing 17-phenyl substitution

Formal name: N-[(2-hydroxy-1-hydroxymethyl)ethyl]-9α,11α,15S-trihydroxy-17-phenyl-18,19,20-trinor-prosta-5Z,13E-dien-1-amide

Synonyms:  17-phenyl trinor PGF2α-SA|Bimatoprost serinol amide

Molecular weight: 461.6

CAS: 1175838-84-2

Purity: ≥98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Neuroscience|Cannabinoid Research|Endocannabinoids

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