An analog of fluprostenol 2-glyceryl ester with increased stability

Fluprostenol serinol amide – 5 mg

Brand:
Cayman
CAS:
1176658-85-7
Storage:
-20
UN-No:
De Minimis - 1170 / 3

2-arachidonyl glycerol (2-AG) exhibits cannabinoid (CB) agonist activity at the CB1 receptor,{5306} is an important endogenous monoglyceride species,{6819} and is thus considered to be the natural ligand for the CB1 receptor. 2-AG can also be metabolized by cyclooxygenase-2 and specific prostaglandin H2 (PGH2) isomerases to form PG 2-glyceryl esters.{11045} Fluprostenol serinol amide (Flu-SA) is a stable analog of PGF2α 2-glyceryl ester that has much greater stability. The biological activity of Flu-SA has not yet been determined.  

 

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SKU: 10004236 - 5 mg Category:

Description

An analog of fluprostenol 2-glyceryl ester with increased stability

Formal name: N-[(2-hydroxy-1-hydroxymethyl)ethyl]-9α,11α,15R-trihydroxy-16-(3-trifluoromethyl)phenoxy)-17,18,19,20-tetranor-prosta-5Z,13E-dien-1-amide

Synonyms:  Flu-SA

Molecular weight: 531.6

CAS: 1176658-85-7

Purity: ≥98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Neuroscience|Cannabinoid Research|Endocannabinoids||Research Area|Neuroscience|Ophthalmology

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